By Jarkko Rautio

This topical reference and guide addresses the chemistry, pharmacology, toxicology and the patentability of prodrugs, completely mirroring the built-in technique popular in cutting-edge drug layout. It summarizes present stories and techniques for the rational layout of prodrugs, starting on the early levels of the improvement strategy, in addition to discussing organ- and site-selective prodrugs.
each corporation utilizing medicinal chemists should be drawn to this practice-oriented assessment of a key technique in smooth drug discovery and development.

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Prodrugs and Targeted Delivery: Towards Better ADME Properties, Volume 47 (Methods and Principles in Medicinal Chemistry) by Jarkko Rautio

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